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Tocris Bioscience™ LEI 101 hydrochloride
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Catalog No. 582610
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10 mg
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Catalog No. Quantity
58-261-0 10 mg
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Catalog No. 58-261-0 Supplier Tocris Bioscience™ Supplier No. 5826/10
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Description

Potent and selective CB2 partial agonist; orally biovailable

Potent and selective CB2 partial agonist (pEC50 = 8.0). Exhibits >100-fold selectivity for CB2 over CB1 and no significant interaction with hFAAH, MAGL, DAGL or NAPE-PLD. Displays antinociceptive activity in a rat neuropathic pain model and attenuates renal inflammation in a mouse kidney damage model. Orally bioavailable with low brain penetration.

Chemical Identifiers

CAS 2250025-91-1

Specifications

Quantity 10 mg
Solubility Soluble to 100mM in DMSO
Formula Weight 508.99
Physical Form Solid
Purity >98%
Chemical Name or Material 3-Cyclopropyl-1-[[4-[6-[(1,1-dioxido-4-thiomorpholinyl)methyl]-5-fluoro-2-pyridinyl]phenyl]methyl]-2

Safety and Handling

Recommended Storage Store at -20°C
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