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  7. Org 27569, Tocris Bioscience™

Org 27569, Tocris Bioscience™

Catalog No. 295750
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Quantity:
10 mg
50 mg
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This item is not returnable. View return policy

Description

Potent allosteric modulator of CB1 receptors

Potent CB1 receptor allosteric modulator (pEC50 = 8.24). Significantly increases binding of the CB1 agonist [3H]CP 55.940 (pKb = 5.67) and decreases binding of the CB1 inverse agonist [3H]SR 141716A (pKb = 5.95). Inhibits CB1 receptor antagonist efficacy in vitro (pKb = 7.57).

Chemical Identifiers

CAS 868273-06-7
Molecular Formula C24H28ClN3O
Molecular Weight (g/mol) 409.96
MDL Number MFCD11045300
InChI Key AHFZDNYNXFMRFQ-UHFFFAOYSA-N
Synonym 5-chloro-3-ethyl-n-4-piperidin-1-yl phenethyl-1h-indole-2-carboxamide, 5-chloro-3-ethyl-1h-indole-2-carboxylic acid 2-4-piperidin-1-yl phenylethyl amide, 5-chloro-3-ethyl-n-2-4-piperidin-1-yl phenyl ethyl-1h-indole-2-carboxamide, d05qtx, org hplc, 5-chloro-3-ethyl-1h-indole-2-carboxylic acid 2-4-piperidin-1-ylphenyl ethyl amide, 5-chloro-3-ethyl-n-2-4-piperidin-1-ylphenyl ethyl-1h-indole-2-carboxamide, 5-chloro-3-ethyl-n-2-4-1-piperidinyl phenyl ethyl-1h-indole-2-carboxamide
PubChem CID 44828492
IUPAC Name 5-chloro-3-ethyl-N-{2-[4-(piperidin-1-yl)phenyl]ethyl}-1H-indole-2-carboxamide
SMILES CCC1=C(NC2=CC=C(Cl)C=C12)C(=O)NCCC1=CC=C(C=C1)N1CCCCC1

Specifications

Quantity 50 mg
Formula Weight 409.95
Percent Purity >99%
Chemical Name or Material Org 27569

Safety and Handling

Recommended Storage Store at Room Temperature
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