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Tocris Bioscience™ OTX 015
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Catalog No. 618110
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61-811-0 10 mg
61-815-0 50 mg
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Catalog No. 61-811-0 Supplier Tocris Bioscience™ Supplier No. 6181/10
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Description

BET bromodomain inhibitor; orally bioavailable

BET bromodomain inhibitor (IC50 values are in the range 92 - 112 nM). Inhibits proliferation and induces apoptosis of leukemia cell lines in vitro. Decreases BRD2, BRD4 and c-MYC protein expression. Orally bioavailable.

Chemical Identifiers

CAS 202590-98-5
Molecular Formula C25H22ClN5O2S

Specifications

Quantity 10 mg
Solubility Soluble to 100mM in DMSO and to 20mM in ethanol
Formula Weight 491.99
Physical Form Solid
Purity >98%
Molecular Weight (g/mol) 491.99
Chemical Name or Material (6S)-4-(4-Chlorophenyl)-N-(4-hydroxyphenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1

Safety and Handling

Recommended Storage Store at -20°C
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