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  5. Tocris Bioscience™ PSB CB5

Tocris Bioscience™ PSB CB5
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Catalog No. 637210
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63-721-0 10 mg
63-725-0 50 mg
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Catalog No. 63-721-0 Supplier Tocris Bioscience™ Supplier No. 6372/10
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Description

Selective GPR18 antagonist

PSB CB5 is a selective GPR18 antagonist (IC50 = 0.279 μM). Exhibits >36-fold selectivity versus CB1 and GPR55 and 14-fold selectivity versus CB2 receptors. Inhibits N-Arachidonylglycine (Cat. No. 1445) induced acrosomal exocytosis in human spermatozoa.

Specifications

Chemical Name or Material (2 Z)-2 [[3-[(4-Chlorophenyl)methoxy]phenyl]methylene]-6,7-dihydro-5 H-imidazo[2,1-b][1,3 ]thiazin-3(2 H)-one
CAS 1627710-30-8
Quantity 10 mg
Target Additional Cannabinoid-related Compounds
Molecular Formula C20H17ClN2O2S
Formula Weight 2020
Purity 98%
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