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  5. Tocris Bioscience™ AZ 191

Tocris Bioscience™ AZ 191
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Catalog No. 523250
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523210 10 mg
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Catalog No. 523250 Supplier Tocris Bioscience™ Supplier No. 5232/50
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Description

Potent DYRK1B inhibitor

AZ 191 is a potent DYRK1B inhibitor (IC50 values are 17, 88 and 1890 nM for DYRK1B, DYRK1A and DYRK2 respectively). Inhibits DYRK1B-induced Gi phase cell cycle arrest in Panc-1 cells in vitro.

Specifications

Chemical Name or Material AZ 191
CAS 1594092-37-1
Synonym N-[2-Methoxy-4-(4-methyl-1-piperazinyl)phenyl]-4-(1-methyl-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-pyrimidinamine
Quantity 50 mg
Solubility Soluble to 100mM in DMSO and to 20mM in ethanol
Molecular Formula C24H27N7O
Formula Weight 429.52
Physical Form Solid
Product Type Bioactive Small Molecule
Purity >98%

Research Use Only. Not For Human or Veterinary Use

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