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Selexipag

Catalog No. 335150
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Quantity:
10 mg
50 mg
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This item is not returnable. View return policy

Description

Selective prostacyclin IP1 receptor agonist

6243Selective prostacyclin IP1 receptor agonist (Ki values are 260 and 2100 nM and for human and rat IP receptors, and >10 μM for EP1-4, DP, FP, and TP receptors). Prodrug for the active form of MRE 269. Ameliorates vascular endothelial dysfunction and increases femoral skin blood flow in rats. Orally available.

Chemical Identifiers

CAS 475086-01-2
Molecular Formula C26H32N4O4S
Molecular Weight (g/mol) 496.63
MDL Number MFCD10567093
InChI Key QXWZQTURMXZVHJ-UHFFFAOYSA-N
Synonym selexipag, uptravi, unii-5exc0e384l, 2-4-5,6-diphenylpyrazin-2-yl isopropyl amino butoxy-n-methylsulfonyl acetamide, 2-4-5,6-diphenylpyrazin-2-yl propan-2-yl amino butoxy-n-methanesulfonyl acetamide, 2-4-n-5,6-diphenylpyrazin-2-yl-n-isopropylamino butyloxy-n-methylsulfonyl acetamide, selexipag usan:inn, uptravi tn, ns-304 selexipag
PubChem CID 9913767
IUPAC Name 2-{4-[(5,6-diphenylpyrazin-2-yl)(propan-2-yl)amino]butoxy}-N-methanesulfonylacetamide
SMILES CC(C)N(CCCCOCC(=O)NS(C)(=O)=O)C1=CN=C(C2=CC=CC=C2)C(=N1)C1=CC=CC=C1

Specifications

Quantity 50 mg
Formula Weight 496.62
Percent Purity >98%
Chemical Name or Material NS 304

Safety and Handling

Recommended Storage Store at -20°C
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