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  5. Tocris™ SK 609

Tocris™ SK 609

Catalog No. 70395
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25 mg
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Catalog No. Quantity
70-395 5 mg
70-392-5 25 mg
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Catalog No. 70-395 Supplier Tocris™ Supplier No. 7039/5
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Description

Dopamine D3 receptor biased agonist

SK 609 is a dopamine D3 receptor biased agonist. Preferentially signals via the G protein-dependent pathway (EC50 values for G protein and β-arrestin-dependent signaling are 1.1 and 50.2 μM, respectively). Exhibits selectivity for D3 over D2 receptors. Improves motor deficits in rodent Parkinson's disease models and ameliorates L-DOPA (Cat. No. 3788) induced abnormal involuntary movements.

Specifications

Chemical Name or Material 2-chloro-α-methyl-benzenepropanamine hydrochloride
CAS 1092797-77-7
Quantity 5 mg
Target Dopamine D3 Receptor Agonists
Molecular Formula C10H14ClN.HCl
Formula Weight 859
Purity 98%
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