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Trap 101, Tocris Bioscience™ Catalog No.: 250850
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Trap 101, Tocris Bioscience™

Catalog No. 250850
50 mg
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Quantity:
50 mg
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Catalog No. 25-085-0

Supplier: R&D Systems 2508/50

This item is not returnable. View return policy

Description

Potent and selective NOP antagonist; active in vivo

Potent and selective nociceptin/orphanin FQ (NOP) receptor antagonist (pA 2 = 7.75). Displays selectivity for NOP receptors over classical opioid receptors (pK i values are 8.65, 6.60, 6.14 and < 5 for NOP, μ-, κ-, and δ-opioid receptors respectively). Attenuates motor deficits in a rat model of Parkinson's Disease. Active in vivo.

Chemical Identifiers

CAS 1216621-00-9
Molecular Formula C24H36ClN3O2
Molecular Weight (g/mol) 434.021
InChI Key YEVMLMQAMCKVSC-UHFFFAOYSA-N
Synonym trap 101, trap-101 hydrochloride, 1-1-cyclooctylmethyl-1,2,3,6-tetrahydro-5-hydroxymethyl-4-pyridinyl-3-ethyl-1,3-dihydro-2h-benzimidazol-2-one hydrochloride, 1-1-cyclooctylmethyl-5-hydroxymethyl-1,2,3,6-tetrahydropyridin-4-yl-3-ethyl-1h-benzo d imidazol-2 3h-one hydrochloride, 1-1-cyclooctylmethyl-3-hydroxymethyl-5,6-dihydro-2h-pyridin-4-yl-3-ethyl-1,3-benzodiazol-2-one hydrochloride, trap101-hcl, trap-101 hydrochloride hplc , powder, 1-1-cyclooctylmethyl-1,2,3,6-tetrahydro-5-hydroxymethyl-4-pyridinyl-3-ethyl-1,3-dihydro-2hbenzimidazol-2-one hydrochloride
PubChem CID 56972178
IUPAC Name 1-[1-(cyclooctylmethyl)-5-(hydroxymethyl)-3,6-dihydro-2H-pyridin-4-yl]-3-ethylbenzimidazol-2-one;hydrochloride
SMILES CCN1C2=CC=CC=C2N(C1=O)C3=C(CN(CC3)CC4CCCCCCC4)CO.Cl

Specifications

Quantity 50 mg
Formula Weight 434.02
Percent Purity >98%
Chemical Name or Material Trap 101

Product Suggestions

Safety and Handling

Recommended Storage Store at +4°C
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