Organic Acids

Medchemexpress LLC Relamorelin (TFA) | 2863659-22-5 | 99.8% | 905.00 | 25 MG

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Small and/or specialty supplier based on Federal laws and SBA requirements.
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Relamorelin TFA is a pentapeptide ghrelin analog and a selective ghrelin/growth hormone secretagogue receptor (GHSR) agonist with a Ki of 0.42 nM for the GHS-1a receptor. It is centrally penetrant, increases growth hormone levels, and accelerates gastric emptying. This compound has potential for research into cachexia, gastroparesis, and gastric/intestinal dysmobility disorders.

• Pentapeptide ghrelin analog
• Selective ghrelin/growth hormone secretagogue receptor (GHSR) agonist
• Ki of 0.42 nM for GHS-1a receptor
• Centrally penetrant
• Increases growth hormone levels
• Accelerates gastric emptying
• Shows ~3 times greater affinity for GHS-1a (Ki=0.42 nM) than native ghrelin (Ki=1.12 nM)
• 6 times more potent (EC50=0.71 nM) in activating the GHS-1a receptor than native ghrelin (EC50=4.2 nM) in vitro by calcium mobilization
• Solid appearance, white to off-white color
• For research use only.

Medchemexpress LLC Relamorelin (TFA) | 2863659-22-5 | 99.8% | 905.00 | 50 MG

Small and Specialty Supplier Partner
Small and/or specialty supplier based on Federal laws and SBA requirements.
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Relamorelin (TFA) | 2863659-22-5 | 99.8% | 905.00 | 50 MG

Medchemexpress LLC Relamorelin (TFA) | 2863659-22-5 | 99.8% | 905.00 | 100 MG

Small and Specialty Supplier Partner
Small and/or specialty supplier based on Federal laws and SBA requirements.
Learn More

Relamorelin (RM-131) TFA, a pentapeptide ghrelin analog, is a selective ghrelin/growth hormone secretagogue receptor (GHSR) agonist with a Ki of 0.42 nM for the GHS-1a receptor. It is centrally penetrant, increases growth hormone levels, and accelerates gastric emptying. Relamorelin TFA has potential for research into cachexia, gastroparesis, and gastric/intestinal dysmobility disorders.

• Selective ghrelin/growth hormone secretagogue receptor (GHSR) agonist.
• Ki of 0.42 nM for GHS-1a receptor.
• Centrally penetrant.
• Increases growth hormone levels.
• Accelerates gastric emptying.
• Potential for cachexia, gastroparesis, and gastric/intestinal dysmobility disorders research.
• Purity: 99.81%.

Medchemexpress LLC CL2A (TFA) | 2616704-22-2 | 99.5% | 1176.24 | C50H79N9O16 | 5 MG

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Small and/or specialty supplier based on Federal laws and SBA requirements.
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CL2A (TFA) is a pH-sensitive, cleavable PEG8- and triazole-containing PABC-peptide-mc linker for use in antibody-drug conjugate construction. The TFA salt form improves handling and stability and is designed to release payloads under acidic conditions to produce a bystander effect.

• Cleavable linker enabling payload release under acidic conditions.
• PEG8 spacer and triazole moiety for increased solubility and stability.
• Designed for conjugation to antibody cysteine residues via disulfide linkage.
• Available in small research-scale packages for use in ADC development.
• Stable as a powder when stored sealed at 4°C; shipped at room temperature.

eMolecules​ Ambeed / (R)-2-(22-Dimethyl-5-oxo-13-dioxolan-4-yl)acetic acid / 1g / 649269522 / A594473 / / 113278-68-5 / MFCD00211272 / 174.152 / C7H10O5

Ambeed / (R)-2-(22-Dimethyl-5-oxo-13-dioxolan-4-yl)acetic acid / 1g / 649269522 / A594473 / / 113278-68-5 / MFCD00211272 / 174.152 / C7H10O5

eMolecules​ AstaTech / 22-DIFLUORO-2-(FLUOROSULFONYL)ACETIC ACID / 5g / 351646826 / P17348 / 95.000 / 1717-59-5 / MFCD01320807 / 178.080 / C2HF3O4S

AstaTech / 22-DIFLUORO-2-(FLUOROSULFONYL)ACETIC ACID / 5g / 351646826 / P17348 / 95.000 / 1717-59-5 / MFCD01320807 / 178.080 / C2HF3O4S

eMolecules​ AstaTech / BENZOIC ACID 4-(ACETYLAMINO)- METHYL ESTER / 0.25g / 796988864 / L10152 / 98.000 / 17012-22-5 / MFCD00463106 / 193.202 / C10H11NO3

AstaTech / BENZOIC ACID 4-(ACETYLAMINO)- METHYL ESTER / 0.25g / 796988864 / L10152 / 98.000 / 17012-22-5 / MFCD00463106 / 193.202 / C10H11NO3

eMolecules​ Ambeed / (R)-5-(12-Dithiolan-3-yl)pentanoic acid / 5g / 552585828 / A147769 / / 1200-22-2 / [null] / 206.320 / C8H14O2S2

Ambeed / (R)-5-(12-Dithiolan-3-yl)pentanoic acid / 5g / 552585828 / A147769 / / 1200-22-2 / [null] / 206.320 / C8H14O2S2

eMolecules​ Ambeed / (2S2S)-22-(Ethane-12-diylbis(azanediyl))bis(butan-1-ol) / 1mg / 761204861 / A939026 / / 74-55-5 / MFCD00866809 / 204.314 / C10H24N2O2

Ambeed / (2S2S)-22-(Ethane-12-diylbis(azanediyl))bis(butan-1-ol) / 1mg / 761204861 / A939026 / / 74-55-5 / MFCD00866809 / 204.314 / C10H24N2O2