5,7-Dimethoxyflavone is a major component of *Kaempferia parviflora* with diverse biological activities. It exhibits anti-obesity, anti-inflammatory, and antineoplastic effects. This compound acts as an inhibitor of cytochrome P450 (CYP) 3As and is a potent Breast Cancer Resistance Protein (BCRP) inhibitor.
- Exhibits anti-obesity, anti-inflammatory, and antineoplastic effects
- Acts as a potent inhibitor of CYP3A and BCRP
- Inhibits Bcrp1-mediated Sorafenib efflux
- Induces melanogenesis
- Inhibits lipid accumulation and adipocyte differentiation
- Reduces liver CYP3A11 and CYP3A25 protein expression
- Inhibits sarcopenia
- Decreases body weight gain and inhibits fatty liver