Oxazinanes
Cayman Chemical SB-242084 (hydrochloride), Purity: ≥98%, CAS: 1049747-87-6, 5 mg
An antagonist of the 5-HT2C receptor (pKi = 9.0), with at least 100-fold more selectivity over other 5-HT, dopamine, or adrenergic receptors; brain penetrant with significant anxiolytic activity; used extensively in animal research
Aobchem 4 5-Dichloro-2-methyl-2H-1 2 3-triazole | 95% | C3H3Cl2N3 | 250mg
4 5-Dichloro-2-methyl-2H-1 2 3-triazole | 95% | C3H3Cl2N3 | 250mg
c1ccccc1 | 1g | 525307271](https://assets.fishersci.com/TFS-Assets/CCG/product-images/5000493374.jpg-250.jpg)
eMolecules 1225376-02-2 | (R)-2-Phenylmorpholine | J & W PharmLab LLC | MFCD18249849 | 163.220 | C10H13NO | 96.000 | C1CO[C@@H](CN1)c1ccccc1 | 1g | 525307271
(R)-2-Phenylmorpholine | J & W PharmLab LLC | 1225376-02-2 | MFCD18249849 | 163.220 | C10H13NO | 96.000 | C1CO[C@@H](CN1)c1ccccc1 | 1g | 525307271
eMolecules 1201905-61-4 | (E)-1-Ethoxyethene-2-boronic acid pinacol ester | Combi-Blocks | MFCD09998813 | 198.070 | C10H19BO3 | 98.000 | CCO\C=C\B1OC(C)(C)C(C)(C)O1 | 5g | 267161125
(E)-1-Ethoxyethene-2-boronic acid pinacol ester | Combi-Blocks | 1201905-61-4 | MFCD09998813 | 198.070 | C10H19BO3 | 98.000 | CCO\C=C\B1OC(C)(C)C(C)(C)O1 | 5g | 267161125
![Medchemexpress LLC 7H-Pyrazolo[4,3-d]pyrimidin-7-one, 5-(2-ethoxyphenyl)-1,6-dihydro-1-methyl-3-propyl- | 139756-21-1 | 99.8% | 312.37 | 250 MG](https://assets.fishersci.com/TFS-Assets/CCG/product-images/5000451606-logo.png-250.jpg){kind=logo}
Medchemexpress LLC 7H-Pyrazolo[4,3-d]pyrimidin-7-one, 5-(2-ethoxyphenyl)-1,6-dihydro-1-methyl-3-propyl- | 139756-21-1 | 99.8% | 312.37 | 250 MG
PDE5-IN-7 (compound 8) is a selective phosphodiesterase 5 (PDE 5) inhibitor with an IC50 value of 5 nM, while having an IC50 of 300 nM for PDE 1. It can be detected and isolated from Sildenafil derivatives. It is intended for research use only and is not sold to patients.
- Selective phosphodiesterase 5 (PDE 5) inhibitor
- IC50 value of 5 nM for PDE5
- IC50 value of 300 nM for PDE1
- Detected and isolated from Sildenafil derivatives
Medchemexpress LLC Ipatasertib dihydrochloride | 1396257-94-5 | C24H34Cl3N5O2 | 500 MG
Ipatasertib dihydrochloride is a highly selective and ATP-competitive pan-Akt inhibitor. It exhibits significant selectivity for Akt1 over closely related kinases PKA and p70S6K, inhibiting only a few other kinases at higher concentrations.
- Highly selective and ATP-competitive pan-Akt inhibitor
- Inhibits Akt1, Akt2, and Akt3
- Exhibits high selectivity against PKA and p70S6K
- Inhibits only three other kinases by more than 70% at 1 μM concentration in a panel of 230 protein kinases