Aminophenols
Medchemexpress LLC CGP71683 hydrochloride | 192322-50-2 | MFCD07783999 | 99.4% | 512.07 g/mol | C26H30ClN5O2S | 1 ML
CGP71683 hydrochloride is a selective, non-peptide neuropeptide Y (NPY) Y5 receptor antagonist (Ki = 1.3 nM) commonly used in receptor pharmacology and signaling research. It demonstrates substantially reduced activity at Y1 and Y2 receptors and is supplied both as a solid and as a pre-made DMSO solution for ready-to-use assays.
- Selective NPY Y5 receptor antagonist (Ki = 1.3 nM).
- High selectivity over Y1 and Y2 receptors.
- Available as solid or 10 mM solution in DMSO, 1 mL.
- High purity suitable for research applications.
- Intended for receptor pharmacology and signaling studies.
Medchemexpress LLC OATD-02 hydrochloride | 2146132-73-0 | 99.9% | 308.61 g/mol | C12H26BClN2O4 | 10 MG
OATD-02 hydrochloride is the hydrochloride salt form of an orally active, competitive, reversible, noncovalent dual inhibitor of arginase 1 and arginase 2, intended for preclinical cancer research. It is supplied as a high-purity, water-soluble solid suitable for in vitro and in vivo studies.
- High purity: 99.9%.
- White to off-white solid physical form.
- High aqueous solubility: 250 mg/mL in water (may require ultrasonic).
- Dual arginase 1 and 2 inhibitory activity for tumor immunology research.
- Available in small research pack sizes for preclinical use.
Matrix Scientific 1-(4-HYDROXYPHENYL)PIPERAZI-10
1-(4-hydroxyphenyl)piperazine Mf C10h14n2o Mw 178.24 Cas 56621-48-8 Mdl MFCD00066156
Medchemexpress LLC RGX-104 (hydrochloride) | 610318-03-1 | 99.9% | 632.54 | 10 MG
RGX-104 hydrochloride is a small-molecule LXR agonist that modulates innate immunity via transcriptional activation of the ApoE gene. It is for research use only and not sold to patients.
- LXR agonist
- Modulates innate immunity via transcriptional activation of the ApoE gene
- Oral administration significantly suppresses the growth of multiple cancer types (e.g., lung cancer, melanoma, glioblastoma, ovarian, renal cell, triple-negative breast, and colon cancer) in animals with palpable tumors.
- Can cause partial or complete tumor regression in some instances.
Medchemexpress LLC Axc-715 hydrochloride | 2490497-93-1 | 99.5% | C18H26ClN5 | 10MG
AXC-715 hydrochloride is the hydrochloride salt of a small-molecule TLR7/TLR8 dual agonist used for preclinical immunology and oncology research. Supplied for research use only, it is described as an immune adjuvant and has been used in synthesis of antibody-adjuvant conjugates and in vivo antitumor models.
- Dual TLR7/TLR8 agonist activity for immune-modulating studies
- High purity (99.5%) for reproducible experimental results
- Hydrochloride salt form improves aqueous solubility relative to the free base
- Suitable for conjugation and formulation in antibody-adjuvant constructs
- Available in small-scale research quantities for preclinical work
- Storage recommendations provided for solid and solution forms to maintain stability
eMolecules 258331-10-1 | TERT-BUTYL 2-(2-HYDROXYPHENYL)ACETATE | AstaTech | MFCD25019077 | 208.257 | C12H16O3 | 95.000 | CC(C)(C)OC(=O)Cc1ccccc1O | 1g | 335884869
TERT-BUTYL 2-(2-HYDROXYPHENYL)ACETATE | AstaTech | 258331-10-1 | MFCD25019077 | 208.257 | C12H16O3 | 95.000 | CC(C)(C)OC(=O)Cc1ccccc1O | 1g | 335884869
Medchemexpress LLC Csrm617 hydrochloride | 1353749-74-2 | 100.0% | 25 MG
CSRM617 hydrochloride is a selective small-molecule inhibitor of the transcription factor ONECUT2 (OC2). It binds the OC2-HOX domain (Kd 7.43 μM in SPR assays), induces apoptosis in preclinical models, and is supplied as a high-purity solid suitable for in vitro and in vivo studies.
- Selective ONECUT2 inhibitor with documented apoptosis induction.
- High purity: 99.97%.
- Available in multiple solid pack sizes including 25 MG.
- Soluble in DMSO: 100 mg/mL; several in vivo formulation protocols provided.
- Storage: solid at -20°C; solutions at -80°C (6 months) or -20°C (1 month).
Apexbio Technology LLC OTS964 hydrochloride 1338545-07-5 2mg
OTS964 hydrochloride (CAS 1338545-07-5) is a selective inhibitor of T-lymphokine-activated killer cell-originated protein kinase (TOPK) demonstrating an IC50 of 28 nM against its target As a dimethylated derivative of OTS514 OTS964 displays high affinity and selectivity for TOPK a serine/threonine kinase implicated in various human malignancies In vitro OTS964 potently suppresses proliferation of multiple TOPK-positive cancer cell lines (IC50 values ranging from 7 6 to 73 nM) while showing markedly reduced activity in TOPK-negative models In in vivo studies OTS964 administered intravenously to mice bearing LU-99 xenografts resulted in significant tumor growth inhibition without notable toxicity Research applications include studying TOPK-related oncogenic pathways and hematopoietic cell differentiation
Medchemexpress LLC Ly-266,097 hydrochloride | 172895-39-5 | MFCD00949080 | ≥98.0% | 407.3 g/mol | C21H23ClN2O2 · HCl | 100 MG
LY266097 hydrochloride is the hydrochloride salt of LY266097, a selective antagonist of the serotonin 5-HT2B receptor used as a research tool in pharmacology and structural biology studies.
- Selective 5-HT2B receptor antagonist for receptor pharmacology studies.
- Supplied as the hydrochloride salt for improved solubility and handling.
- High purity suitable for in vitro and structural biology applications.
- Available in small research quantities for assay development and screening.