Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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Quantity
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2,266
Tocris Bioscience™ Ro 3306
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CAS: 872573-93-8 Molecular Formula: C18H13N3OS2
| CAS | 872573-93-8 |
|---|---|
| Molecular Formula | C18H13N3OS2 |
2,267
Tocris Bioscience™ Imetit dihydrobromide
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CAS: 32385-58-3 Molecular Formula: C6H12Br2N4S
| CAS | 32385-58-3 |
|---|---|
| Molecular Formula | C6H12Br2N4S |
2,268
Tocris Bioscience™ (-)-Cytisine
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CAS: 485-35-8 Molecular Formula: C11H14N2O
| CAS | 485-35-8 |
|---|---|
| Molecular Formula | C11H14N2O |
2,269
Tocris Bioscience™ AZD 4547
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Potent and selective FGFR inhibitor
| Target | FGF Receptor Inhibitors |
|---|---|
| CAS | 1035270-39-3 |
| Chemical Name or Material | rel-N-[5-[2-(3,5-Dimethoxyphenyl)ethyl]-1H-pyrazol-3-yl]-4-[(3R,5S)-3,5-dimethyl-1-piperazinyl]benzamide |
| Molecular Formula | C26H33N5O3 |
2,270
Tocris Bioscience™ TPEN
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CAS: 16858-02-9 Molecular Formula: C26H28N6
| CAS | 16858-02-9 |
|---|---|
| Molecular Formula | C26H28N6 |
2,271
Tocris Bioscience™ 1R,3R-RSL3
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Negative control for 1S,3R-RSL3 (Cat. No. 6118)
| Target | Glutathione Peroxidase 4/GPX4 |
|---|---|
| CAS | 1219810-15-7 |
| Purity | 0.98 |
| Chemical Name or Material | (1 R,3 R)-Methyl 2-(2-chloroacetyl)-2,3,4,9-tetrahydro-1-[4-(methoxycarbonyl)phenyl]-1 H-pyrido[3,4-b]indole-3-carboxylate |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C23H21ClN2O5 |
2,272
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Tocris Bioscience™ C26-A6
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Tocris Bioscience™ C26-A6
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Disrupts MTDH and SND1 interaction, enhances immune surveillance
| Target | Cell Adhesion Inhibitors |
|---|---|
| CAS | 1341030-00-9 |
| Purity | 0.98 |
| Chemical Name or Material | 5-Chloro-2-methoxy-N-(2-methyl[1,2,4 ]triazolo[1,5-a]pyridin-8-yl)benzenesulfonamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C14H13ClN4O3S |
2,273
Tocris Bioscience™ GSK 2018682
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S1P1 and S1P5 agonist
| Product Type | Agonist |
|---|---|
| Purity | 98% |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C22H21ClN4O4 |
| Formula Weight | 440.88 |
2,274
Tocris Bioscience™ PG 01037 dihydrochloride
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CAS: 675599-62-9 Molecular Formula: C26H28Cl4N4O
| CAS | 675599-62-9 |
|---|---|
| Molecular Formula | C26H28Cl4N4O |
2,275
Tocris Bioscience™ DY 268
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Potent FXR antagonist
| Target | LXR-like Receptor Antagonists |
|---|---|
| CAS | 1609564-75-1 |
| Purity | >98% |
| Chemical Name or Material | 1-[(3-Methoxyphenyl)methyl]-N-[4-methyl-3-(4-morpholinylsulfonyl)phenyl]-3-(4-methylphenyl)-1H-pyrazole-4-carboxamide |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C30H32N4O5S |
| Formula Weight | 560.66 |
2,276
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Tocris Bioscience™ Mesopram
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Tocris Bioscience™ Mesopram
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CAS: 189940-24-7 Molecular Formula: C14H19NO4
| CAS | 189940-24-7 |
|---|---|
| Molecular Formula | C14H19NO4 |
2,277
Tocris Bioscience™ CK 666
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CAS: 442633-00-3 Molecular Formula: C18H17FN2O
| CAS | 442633-00-3 |
|---|---|
| Molecular Formula | C18H17FN2O |
2,278
Tocris Bioscience™ Thalidomide 4'-oxyacetamide-alkylC4-azide
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Azide-functionalized Thalidomide; click cereblon ligand for PROTACs
2,279
Tocris Bioscience™ ML 323
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Potent and selective USP1-UAF1 allosteric inhibitor
| CAS | 1572414-83-5 |
|---|---|
| Purity | 98% |
| Recommended Storage | Store at -20°C |
| Synonym | 5-Methyl-2-[2-(1-methylethyl)phenyl]-N-[[4-(1H-1,2,3-triazol-1-yl)phenyl]methyl]-4-pyrimidinamine |
| Molecular Formula | C23H24N6 |
| Formula Weight | 384.48 |
2,280
Tocris Bioscience™ GYKI 53655 hydrochloride
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CAS: 143692-48-2 Molecular Formula: C19H21ClN4O3
| CAS | 143692-48-2 |
|---|---|
| Molecular Formula | C19H21ClN4O3 |