Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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Molecular Weight (g/mol)
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2,416
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2,416
R&D Systems™ TFB-TBOA
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. High affinity EAAT1 and EAAT2 blocker
| CAS | 480439-73-4 |
|---|---|
| Solubility | Soluble to 100mM in DMSO |
| Chemical Name or Material | (3S)-3-[[3-[[4-(Trifluoromethyl)benzoyl]amino]phenyl]methoxy]-L-aspartic acid |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C19H17F3N2O6 |
| Formula Weight | Observed MW: 426.35 |
| Assay Percent Range | >98% |
2,417
R&D Systems™ TP 472
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent BRD9/7 inhibitor
2,418
R&D Systems™ VH 032 amide-alkylC4-amine
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. PROTACs (Proteolysis Targeting Chimeras)
2,419
R&D Systems™ FITM
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent and selective negative allosteric modulator of mGlu1 receptors
| Product Type | Negative Allosteric Modulator |
|---|---|
| Purity | 98% |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C18H18FN5OS |
| Formula Weight | 371.43 |
2,420
R&D Systems™ GSK 269962
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 850664-21-0 Molecular Formula: C29H30N8O5
| CAS | 850664-21-0 |
|---|---|
| Molecular Formula | C29H30N8O5 |
2,421
R&D Systems™ E-4031 dihydrochloride
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Greener Choice
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 113559-13-0 Molecular Formula: C21H29Cl2N3O3S
| CAS | 113559-13-0 |
|---|---|
| Molecular Formula | C21H29Cl2N3O3S |
2,422
R&D Systems™ SR 57227 hydrochloride
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 77145-61-0 Molecular Formula: C10H15Cl2N3
| CAS | 77145-61-0 |
|---|---|
| Molecular Formula | C10H15Cl2N3 |
2,423
R&D Systems™ Thalidomide 5'-amine-alkylC8-amine
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Cereblon ligand with alkyl linker and terminal amine for onward chemistry
2,424
R&D Systems™ ACET
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 936095-50-0 Molecular Formula: C20H21N3O6S
| CAS | 936095-50-0 |
|---|---|
| Molecular Formula | C20H21N3O6S |
2,425
R&D Systems™ Ivosidenib
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent inhibitor of mutant isocitrate dehydrogenase (mIDH1)
| Target | Isocitrate Dehydrogenase 1/IDH1 |
|---|---|
| CAS | 1448347-49-6 |
| Chemical Name or Material | (2S)-N-{(1S)-1-(2-Chlorophenyl)-2-[(3,3-difluorocyclobutyl)amino]-2-oxoethyl}-1(4-cyanopyridin-2-yl)-N-(5-fluoropyridin-3-yl)-5-oxopyrrolidine-2-carboxamide |
| Recommended Storage | Store the unopened product at -20 to -70 °C. Use a manual defrost freezer and avoid repeated freeze-thaw cycles. Do not use past expiration date. |
| Molecular Formula | C28H22ClF3N6O3 |
2,426
R&D Systems™ GSK2578215A
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. Potent, selective LRRK2 inhibitor; brain penetrant
| CAS | 1285515-21-0 |
|---|---|
| Chemical Name or Material | 5-(2-Fluoro-4-pyridinyl)-2-(phenylmethoxy)-N-3-pyridinylbenzamide |
| Recommended Storage | Store at Room Temperature |
| Molecular Formula | C24H18FN3O2 |
| Formula Weight | Observed MW: 399.42 |
| Assay Percent Range | >99% |
2,427
R&D Systems™ Diclofenac sodium salt
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 15307-79-6 Molecular Formula: C14H10Cl2NNaO2
| CAS | 15307-79-6 |
|---|---|
| Molecular Formula | C14H10Cl2NNaO2 |
2,428
R&D Systems™ PF 04885614
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 1480833-70-2 Molecular Formula: C13H14F3N3O
| CAS | 1480833-70-2 |
|---|---|
| Molecular Formula | C13H14F3N3O |
2,429
R&D Systems™ Bosentan
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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A Tocris product, part of R&D Systems. High affinity dual ETA and ETB receptor antagonist;orally bioavailable
| Target | Non-selective Endothelin Receptor |
|---|---|
| CAS | 147536-97-8 |
| Product Type | Antagonist |
| Recommended Storage | Store at 4°C |
| Molecular Formula | C27H29N5O6S |
| Formula Weight | 551.61g/mol |
2,430
R&D Systems™ 4-IPP
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 41270-96-6 Molecular Formula: C10H7IN2
| CAS | 41270-96-6 |
|---|---|
| Molecular Formula | C10H7IN2 |