Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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436
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450
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436
Tocris Bioscience™ VH 032 amide-alkylC5-amine
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VHL ligand with alkyl linker and terminal amine for onward chemistry
437
Tocris Bioscience™ R 7050
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Inhibitor of TNF-α receptor 1 signaling
| Inhibitors | R 7050 |
|---|---|
| Product Type | R 7050 |
| Molecular Weight (g/mol) | 380.77 |
| Purity | >98% |
438
Tocris Bioscience™ BIO
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CAS: 667463-62-9 Molecular Formula: C16H10BrN3O2
| CAS | 667463-62-9 |
|---|---|
| Molecular Formula | C16H10BrN3O2 |
439
Tocris Bioscience™ PF 04885614
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CAS: 1480833-70-2 Molecular Formula: C13H14F3N3O
| CAS | 1480833-70-2 |
|---|---|
| Molecular Formula | C13H14F3N3O |
440
Tocris Bioscience™ MRTX 849
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Mutation-selective inhibitor of KRASG12C
| Target | Ras GTPase Inhibitors |
|---|---|
| CAS | 2326521-71-3 |
| Purity | 98% |
| Chemical Name or Material | 4-[7-(8-Chloro-1-naphthalenyl)-5,6,7,8-tetrahydro-2-[[(2 S)-1-methyl-2-pyrrolidinyl]methoxy]pyrido[3,4-d]pyrimidin-4-yl]-1-(2-fluoro-1-oxo-2-propen-1-yl)-(2 S)-2-piperazineacetonitrile |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C32H35ClFN7O2 |
441
Tocris Bioscience™ Ro 5-3335
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Core binding factor inhibitor; attenuates hematopoiesis
442
Tocris Bioscience™ Laropiprant
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Potent and selective prostaglandin D2 receptor antagonist
| Target | Prostanoid Receptor Antagonists |
|---|---|
| CAS | 571170-77-9 |
| Purity | 0.98 |
| Chemical Name or Material | (3 R)-4-[(4-Chlorophenyl)methyl]-7-fluoro-1,2,3,4-tetrahydro-5-(methylsulfonyl)cyclopent[b]indole-3-acetic acid |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C21H19ClFNO4S |
443
Tocris Bioscience™ NS 8593 Hydrochloride
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Selective negative modulator of KCa2 (SK) channels; inhibits SK currents
| CAS | 875755-24-1 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 100mM in DMSO and to 20mM in ethanol |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | NS 8593 hydrochloride |
| Recommended Storage | Store at 4°C |
| Synonym | N-[(1R)-1,2,3,4-Tetrahydro-1-naphthalenyl]-1H-benzimidazol-2-amine hydrochloride |
| Molecular Formula | C17H17N3·HCl |
| Formula Weight | 299.8 |
445
Tocris Bioscience™ GR 55562 dihydrochloride
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 159533-25-2 Molecular Formula: C23H27Cl2N3O2
| CAS | 159533-25-2 |
|---|---|
| Molecular Formula | C23H27Cl2N3O2 |
446
Tocris Bioscience™ SIS3
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Selective Smad3 inhibitor; inhibits TGF-βR1 signaling
| Product Type | SIS3 |
|---|---|
| Molecular Weight (g/mol) | 489.99 |
| Purity | 97% |
447
Tocris Bioscience™ Bupropion hydrochloride
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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CAS: 31677-93-7 Molecular Formula: C13H19Cl2NO
| CAS | 31677-93-7 |
|---|---|
| Molecular Formula | C13H19Cl2NO |
448
Tocris Bioscience™ AZ 12799734
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent TGF-βRI inhibitor
| CAS | 1117684-36-2 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 4-[[4-[(2.6-Dimethyl-3-pyridinyl)oxy]-2-pyridinyl]amino]benzenesulfonamide |
| Molecular Formula | C18H18N4O3S |
449
Tocris Bioscience™ GPR52 Comp-43
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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GPR52 receptor antagonist
| Target | Orphan 7-TM Receptor Antagonists |
|---|---|
| CAS | 1239987-91-7 |
| Purity | 0.98 |
| Chemical Name or Material | (2 E)-5-Phenyl-1-(2-thienyl)-2-penten-1-one |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C15H14OS |
450
Tocris Bioscience™ L-690,330
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CAS: 142523-38-4 Molecular Formula: C8H12O8P2
| CAS | 142523-38-4 |
|---|---|
| Molecular Formula | C8H12O8P2 |