Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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1
| CAS | 160003-66-7 |
|---|---|
| Molecular Formula | C7 H5 I N2 O3 |
2
| CAS | 10605-02-4 |
|---|---|
| Molecular Formula | C21 H22 Cl N O4 |
3
Invitrogen™ Nile Red
For use with fluorescence microscopy
Encompass Procurement Services
Non-distribution item offered as a customer accommodation; additional freight charges may apply.
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Non-distribution item offered as a customer accommodation; additional freight charges may apply.
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4
Tocris Bioscience™ CU-T12-9
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent TLR1/2 agonist
| CAS | 1821387-73-8 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 100mM in DMSO and to 20mM in ethanol |
| Purity | >99% |
| Physical Form | Solid |
| Chemical Name or Material | CU-T12-9 |
| Recommended Storage | Store at 4°C |
| Synonym | N-Methyl-4-nitro-2-(4-(4-trifluoromethyl)phenyl)-1H-imidazol-1-yl)aniline |
| Molecular Formula | C17H13F3N4O2 |
| Formula Weight | 362.31 |
5
Tocris Bioscience™ Edaglitazone
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and selective PPARγ agonist; antidiabetic
| CAS | 213411-83-7 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 100mM in DMSO |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | Edaglitazone |
| Recommended Storage | Store at 4°C |
| Synonym | 5-[[4-[2-(5-Methyl-2-phenyl-4-oxazolyl)ethoxy]benzo[b]thien-7-yl]methyl]-2,4-thiazolidinedione |
| Molecular Formula | C24H20N2O4S2 |
| Formula Weight | 464.56 |
6
Tocris Bioscience™ TC-I 2014
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent TRPM8 antagonist
| CAS | 1221349-53-6 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 100mM in DMSO and to 100mM in ethanol |
| Purity | >98% |
| Physical Form | Powder |
| Chemical Name or Material | TC-I 2014 |
| Recommended Storage | Store at 4°C |
| Synonym | 3-[7-(Trifluoromethyl)-5-[2-(trifluoromethyl)phenyl]-1H-benzimidazol-2-yl]-1-oxa-2-azaspiro[4.5]dec-2-ene |
| Molecular Formula | C23H19F6N3O |
| Formula Weight | 467.41 |
7
Tocris Bioscience™ ASP 7663
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Selective TRPA1 activator
| CAS | 1190217-35-6 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 100mM in DMSO and to 100mM in ethanol |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | ASP 7663 |
| Recommended Storage | Store at 4°C |
| Synonym | (2E)-2-[7-Fluoro-1,2-dihydro-1-(2-methylpropyl)-2-oxo-3H-indol-3-ylidene]acetic acid |
| Molecular Formula | C14H14FNO3 |
| Formula Weight | 263.26 |
8
Tocris Bioscience™ AZ 191
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent DYRK1B inhibitor
| CAS | 1594092-37-1 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 100mM in DMSO and to 20mM in ethanol |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | AZ 191 |
| Recommended Storage | Store at -20°C |
| Synonym | N-[2-Methoxy-4-(4-methyl-1-piperazinyl)phenyl]-4-(1-methyl-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-pyrimidinamine |
| Molecular Formula | C24H27N7O |
| Formula Weight | 429.52 |
9
Tocris Bioscience™ ONO 8130
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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EP1 receptor antagonist
| CAS | 459841-96-4 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 100mM in DMSO and to 20mM in ethanol |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | ONO 8130 |
| Recommended Storage | Store at 4°C |
| Synonym | 4-[[[2,3-Dihydro-6-[(2-methylpropyl)[(4-methyl-2-thiazolyl)sulfonyl]amino]-1H-indene-5yl]oxy]methyl]benzoic acid |
| Molecular Formula | C25H28N2O5S2 |
| Formula Weight | 500.63 |
10
Tocris Bioscience™ Cerestat
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and noncompetitive NMDA receptor antagonist
| CAS | 137160-11-3 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 50mM in water and to 100mM in DMSO |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | Cerestat |
| Recommended Storage | Store at 4°C |
| Synonym | N-(3-Ethylphenyl)-N-methyl-N'-1-naphthalenylguanidine hydrochloride |
| Molecular Formula | C20H21N3·HCl |
| Formula Weight | 339.86 |
11
Tocris Bioscience™ ESI 09
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Epac inhibitor
| CAS | 263707-16-0 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 100mM in DMSO and to 20mM in ethanol |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | EPAC Inhibitors |
| Recommended Storage | Store at 4°C |
| Synonym | α-[(2-(3-Chlorophenyl)hydrazinylidene]-5-(1,1-dimethylethyl)-β-oxo-3-isoxazolepropanenitrile |
| Molecular Formula | C16H15ClN4O2 |
| Formula Weight | 330.77 |
12
Tocris Bioscience™ ABT 089 Dihydrochloride
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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High affinity and selective α4β2 nAChR partial agonist
| CAS | 161416-61-1 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 100mM in water and to 20mM in DMSO |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | ABT 089 dihydrochloride |
| Recommended Storage | Desiccate at Room Temperature |
| Synonym | 2-Methyl-3-[(2S)-pyrrolidinylmethoxy]pyridine dihydrochloride |
| Molecular Formula | C11H16N2O·2HCl |
| Formula Weight | 265.18 |
13
Tocris Bioscience™ OICR 9429
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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High affinity and selective WDR5 antagonist
| Target | Additional Lysine Methyltransferase Compounds |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 50mM in DMSO |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | OICR 9429 |
| Recommended Storage | Store at -20°C |
| Synonym | N-[2-(4-Methylpiperazin-1-yl)-5-[3-(morpholin-4-ylmethyl)phenyl]phenyl]-6-oxo-4-(trifluoromethyl)-1,6-dihydropyridine-3-carboxamide |
| Molecular Formula | C29H32F3N5O3 |
| Formula Weight | 555.59 |
14
Tocris Bioscience™ PFK 15
Greener Choice
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Selective PFKFB3 inhibitor
| CAS | 4382-63-2 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 100mM in DMSO |
| Purity | >99% |
| Physical Form | Solid |
| Chemical Name or Material | PFK 15 |
| Recommended Storage | Store at -20°C |
| Synonym | 1-(4-Pyridinyl)-3-(2-quinolinyl)-2-propen-1-one |
| Molecular Formula | C17H12N2O |
| Formula Weight | 260.29 |
15
Tocris Bioscience™ C16
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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PKR inhibitor
| CAS | 608512-97-6 |
|---|---|
| Product Type | Bioactive Small Molecule |
| Solubility | Soluble to 50mM in DMSO and to 20mM in ethanol |
| Purity | >98% |
| Physical Form | Solid |
| Chemical Name or Material | C16 |
| Recommended Storage | Store at -20°C |
| Synonym | 6,8-Dihydro-8-(1H-imidazol-5-ylmethylene)-7H-pyrrolo[2,3-g]benzothiazol-7-one |
| Molecular Formula | C13H8N4OS |
| Formula Weight | 268.29 |