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Tocris Bioscience™ ABT 639
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Catalog No. 677010
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67-701-0 10 mg
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Catalog No. 67-701-0 Supplier Tocris Bioscience™ Supplier No. 6770/10
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Description

CaV3.2 and CaV3.1 channel blocker (IC50 = 2.3 μM)

ABT 639 is a CaV3.2 channel blocker (IC50 = 2.3 μM). Also blocks low voltage-activated (CaV3.1) currents in native rat DRG neurons (IC50 = 7.6 μM). Exhibits little or no activity at other ion channels and receptors. Displays antinociceptive effects in a mechanical hyperalgesia model in vivo. Orally bioavailable.

Specifications

Chemical Name or Material 4-Chloro-2-fluoro-N-(2-fluorophenyl)-5-[[(8aR)-hexahydropyrrolo[1,2-a]pyrazin-2(1H)-yl]carbonyl]benzenesulfonamide
CAS 1235560-28-7
Quantity 10 mg
Molecular Formula C20H20ClF2N3O3S
Formula Weight 455.91
Purity 98%
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