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  9. AM 251, Tocris Bioscience™ 

AM 251, Tocris Bioscience™ Available on GSA/VA Contract for Federal Government customers only.

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50mg
This item is not returnable. View return policy
183232-66-8
C22H21Cl2IN4O
555.241
BUZAJRPLUGXRAB-UHFFFAOYSA-N
unii-3i4fa44mai,1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-piperidin-1-yl-1h-pyrazole-3-carboxamide,n-piperidin-1-yl-5-4-iodophenyl-1-2,4-dichlorophenyl-4-methyl-1h-pyrazole-3-carboxamide,3i4fa44mai,1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-piperidin-1-ylpyrazole-3-carboxamide,n-piperidin-1-yl-5-4-iodophenyl-1-2, 4-dichlorophenyl-4-methyl-1h-pyrazole-3-carboxamide,1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-1-piperidinyl-1h-pyrazole-3-carboxamide,am 251 pharmaceutical,tocris-1117,d08yqt
2125
1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-piperidin-1-ylpyrazole-3-carboxamide
CC1=C(N(N=C1C(=O)NN2CCCCC2)C3=C(C=C(C=C3)Cl)Cl)C4=CC=C(C=C4)I
This item is not returnable. View return policy
183232-66-8
C22H21Cl2IN4O
555.241
BUZAJRPLUGXRAB-UHFFFAOYSA-N
unii-3i4fa44mai,1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-piperidin-1-yl-1h-pyrazole-3-carboxamide,n-piperidin-1-yl-5-4-iodophenyl-1-2,4-dichlorophenyl-4-methyl-1h-pyrazole-3-carboxamide,3i4fa44mai,1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-piperidin-1-ylpyrazole-3-carboxamide,n-piperidin-1-yl-5-4-iodophenyl-1-2, 4-dichlorophenyl-4-methyl-1h-pyrazole-3-carboxamide,1-2,4-dichlorophenyl-5-4-iodophenyl-4-methyl-n-1-piperidinyl-1h-pyrazole-3-carboxamide,am 251 pharmaceutical,tocris-1117,d08yqt
2125
1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-piperidin-1-ylpyrazole-3-carboxamide
CC1=C(N(N=C1C(=O)NN2CCCCC2)C3=C(C=C(C=C3)Cl)Cl)C4=CC=C(C=C4)I

Description

Potent CB1 antagonist; also GPR55 agonist

Potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 306-fold selectivity over CB2 receptors. Also potent GPR55 agonist (EC50 = 39 nM) and μ-opioid receptor antagonist (Ki = 251 nM).

Fluorescent Form also available.

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Quantity 1mg
Formula Weight 555.24
Percent Purity >99%
Chemical Name or Material AM 251

Safety and Handling

Recommended Storage : Store at Room Temperature