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  5. Tocris Bioscience™ AM 251

Tocris Bioscience™ AM 251

Catalog No. 11171
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Catalog No. Quantity
11-171 1 mg
11-171-0 10 mg
11-175-0 50 mg
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Catalog No. 11-171 Supplier Tocris Bioscience™ Supplier No. 1117/1
This item is not returnable. View return policy

Description

Potent CB1 antagonist; also GPR55 agonist

Potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 306-fold selectivity over CB2 receptors. Also potent GPR55 agonist (EC50 = 39 nM) and μ-opioid receptor antagonist (Ki = 251 nM).

Fluorescent Form also available.

Chemical Identifiers

CAS 183232-66-8
Molecular Formula C22H21Cl2IN4O

Specifications

Quantity 1 mg
Formula Weight 555.24
Purity >99%
Molecular Weight (g/mol) 555.241
Chemical Name or Material AM 251

Safety and Handling

Recommended Storage Store at Room Temperature
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