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Tocris Bioscience™ AR-C 118925XX
Selective and competitive P2Y2 antagonist
Supplier: Tocris Bioscience™ 4890/5
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Description
AR-C 118925XX is a potent, selective, competitive and reversible P2Y2 receptor antagonist (pA2 = 8.43). Inactive against a panel of 37 other receptors at a concentration of 10 μM. AR-C 118925XX inhibits ATP-γS-induced mucin secretion in bronchial epithelial cells (IC50 = 1 μM). Inhibits P2Y2 receptor-induced β-arrestin translocation in vitro (pA2 = 37.2-51.3 nM).Specifications
| 5-[[5-(2,8-Dimethyl-5H-dibenzo[a,d]cyclohepten-5-yl)-3,4-dihydro-2-oxo-4-thioxo-1(2H)-pyrimidinyl]methyl]-N-2H-tetrazol-5-yl-2-furancarboxamide | |
| 5 mg | |
| C28H23N7O3S | |
| >98% |
| 216657-60-2 | |
| P2Y Receptor Antagonists | |
| 537.59 |
Safety and Handling
Recommended Storage : Store at -20°C
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