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Tocris Bioscience™ AR-C 118925XX
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Catalog No. 48905
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48-905 5 mg
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Catalog No. 48-905 Supplier Tocris Bioscience™ Supplier No. 4890/5
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Description

Selective and competitive P2Y2 antagonist

AR-C 118925XX is a potent, selective, competitive and reversible P2Y2 receptor antagonist (pA2 = 8.43). Inactive against a panel of 37 other receptors at a concentration of 10 μM. AR-C 118925XX inhibits ATP-γS-induced mucin secretion in bronchial epithelial cells (IC50 = 1 μM). Inhibits P2Y2 receptor-induced β-arrestin translocation in vitro (pA2 = 37.2-51.3 nM).

Specifications

Chemical Name or Material 5-[[5-(2,8-Dimethyl-5H-dibenzo[a,d]cyclohepten-5-yl)-3,4-dihydro-2-oxo-4-thioxo-1(2H)-pyrimidinyl]methyl]-N-2H-tetrazol-5-yl-2-furancarboxamide
CAS 216657-60-2
Quantity 5 mg
Target P2Y Receptor Antagonists
Molecular Formula C28H23N7O3S
Formula Weight 537.59
Purity >98%
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