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Tocris Bioscience™ AZ 6102
Potent TNKS1/2 inhibitor
Supplier: Tocris Bioscience™ 5775/50
This item is not returnable.
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Description
AZ 6102 is a potent TNKS2 and TNKS1 inhibitor (IC50 values are 1 and 3 nM, respectively). Exhibits >100-fold selectivity for TNKS1/2 over PARP-1, PARP-2 and PARP-6. Inhibits Wnt signaling in DLD-1 cells (IC50 = 5 nM). Exhibits moderate oral bioavailability.Specifications
| rel-2-[4-[6-[(3R,5S)-3,5-Dimethyl-1-piperazinyl]-4-methyl-3-pyridinyl]phenyl]-3,7-dihydro-7-methyl-4H-pyrrolo[2,3-d]pyrimidin-4-one | |
| 50 mg | |
| C25H28N6O | |
| >98% |
| 1645286-75-4 | |
| Tankyrase Inhibitors | |
| 428.53 |
Safety and Handling
Recommended Storage : Store at -20°C
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