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Tocris Bioscience™ BI 9564
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Catalog No. 559010
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10 mg
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55-901-0 10 mg
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Catalog No. 55-901-0 Supplier Tocris Bioscience™ Supplier No. 5590/10
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Description

Potent and selective BRD9 and BRD7 inhibitor; orally active

BI 9564 is a potent and selective BRD9 and BRD7 inhibitor (Kd values are 14 and 239 nM, respectively). Exhibits selectivity for BRD9/7 over 48 other bromodomains, 324 kinases and 55 GPCRs. Inhibits proliferation of AML cell lines in vitro and reduces AML tumor xenograft growth in vivo. Cell permeable and orally active.

Specifications

Chemical Name or Material 4-[4-[(Dimethylamino)methyl]-2,5-dimethoxyphenyl]-2-methyl-1,2-dihydro-2,7-naphthyridin-1-one
CAS 1883429-22-8
Quantity 10 mg
Target Bromodomain Inhibitors
Molecular Formula C20H23N3O3
Formula Weight 353.41
Purity >98%
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