Promotional price valid on web orders only. Your contract pricing may differ. Interested in signing up for a dedicated account number?
Learn More
  1. Home
  2. Products
  3. Protein Analysis Reagents
  4. Bioactive Small Molecules
  5. Tocris Bioscience™ BIIE 0246 hydrochloride

Tocris Bioscience™ BIIE 0246 hydrochloride
GREENER_CHOICE

Catalog No. 737710
Change view
Click to view available options
Quantity:
1 mg
10 mg
2 product options available for selection
Product selection table with 2 available options. Use arrow keys to navigate and Enter or Space to select.
Catalog No. Quantity
73-771-0 10 mg
RD73771 1 mg
Use arrow keys to navigate between rows. Press Enter or Space to select a product option. 2 options available.
2 options
This item is not returnable. View return policy
Catalog No. 73-771-0 Supplier Tocris Bioscience™ Supplier No. 7377/10
Only null left
Add to Cart
Add to Cart
This item is not returnable. View return policy

Description

Potent, selective and competitive non-peptide NPY Y2 receptor antagonist; active in vivo

BIIE 0246 hydrochloride is a potent, selective and competitive nonpeptide antagonist for the neuropeptide Y Y2 receptor (IC50 = 15 nM). Displays > 650-fold selectivity for NPY Y2 over Y1, Y4 and Y5 receptors. Active in vivo.

Specifications

Chemical Name or Material N-[(1 S)-4-[(Aminoiminomethyl)amino]-1-[[[2-(3,5-dioxo-1,2-diphenyl-1,2,4-triazolidin-4-yl)ethyl]amino]carbonyl]butyl]-1-[2-[4-(6,11-dihydro-6-oxo-5 H-dibenz[b,e]azepin-11-yl)-1-piperazinyl]-2-oxoethyl]-cyclopentaneacetamide hydrochloride
CAS 2624332-04-1
Quantity 10 mg
Target NPY Receptor Antagonists
Molecular Formula C49H57N11O6.HCl
Purity 0.98
Product Title
Select an issue

By clicking Submit, you acknowledge that you may be contacted by Fisher Scientific in regards to the feedback you have provided in this form. We will not share your information for any other purposes. All contact information provided shall also be maintained in accordance with our Privacy Policy.