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CGP 78608 hydrochloride, Tocris Bioscience™

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Quantity:
10mg
50mg
This item is not returnable. View return policy
1135278-54-4
C11H14BrClN3O5P
414.577
MZQQZBPMRPDKTB-JEDNCBNOSA-N
cgp 78608 hydrochloride, 1s-n-7-bromo-2,3-dioxo-1,2,3,4-tetrahydroquinoxalin-5-yl methyl-1-phosphonoethanaminium chloride, 1s-1-7-bromo-2,3-dioxo-1,2,3,4-tetrahydroquinoxalin-5-yl methyl amino ethyl phosphonic acid hydrochloride, pamqx, 1s-1-7-bromo-1,2,3,4-tetrahydro-2,3-dioxo-5-quinoxalinyl methyl amino ethyl phosphonic acid hydrochloride
24978530
CHEBI:64065
[(1S)-1-[(7-bromo-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)methylamino]ethyl]phosphonic acid;hydrochloride
CC(NCC1=CC(=CC2=C1NC(=O)C(=O)N2)Br)P(=O)(O)O.Cl
This item is not returnable. View return policy
1135278-54-4
C11H14BrClN3O5P
414.577
MZQQZBPMRPDKTB-JEDNCBNOSA-N
cgp 78608 hydrochloride, 1s-n-7-bromo-2,3-dioxo-1,2,3,4-tetrahydroquinoxalin-5-yl methyl-1-phosphonoethanaminium chloride, 1s-1-7-bromo-2,3-dioxo-1,2,3,4-tetrahydroquinoxalin-5-yl methyl amino ethyl phosphonic acid hydrochloride, pamqx, 1s-1-7-bromo-1,2,3,4-tetrahydro-2,3-dioxo-5-quinoxalinyl methyl amino ethyl phosphonic acid hydrochloride
24978530
CHEBI:64065
[(1S)-1-[(7-bromo-2,3-dioxo-1,4-dihydroquinoxalin-5-yl)methylamino]ethyl]phosphonic acid;hydrochloride
CC(NCC1=CC(=CC2=C1NC(=O)C(=O)N2)Br)P(=O)(O)O.Cl

Potent, selective glycine-site NMDA antagonist

Potent and selective NMDA antagonist that acts through the glycine site (IC50 = 5 nM). Displays > 500-fold selectivity over kainate and AMPA receptors (IC50 values are 2.7 and 3 μM respectively). Also potentiates GluN1/GluN3A-mediated glycine currents (EC50 = 26.3 nM). Anticonvulsant in vivo following systemic administration.
Quantity 50mg
Formula Weight 414.58
Percent Purity >98%
Chemical Name or Material CGP 78608 hydrochloride

Recommended Storage : Store at Room Temperature