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Tocris Bioscience™ CID 16020046
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Catalog No. 495925
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25 mg
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Catalog No. Quantity
49-592-5 25 mg
49-595 5 mg
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Catalog No. 49-592-5 Supplier Tocris Bioscience™ Supplier No. 4959/25
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Description

Selective GPR55 antagonist

CID 16020046 is a selective GPR55 antagonist. Inhibits LPI-induced Ca2+ signaling (IC50 = 0.21 μM in HEK-GPR55 cells), ERK1/2 phosphorylation and GPR55-mediated transcription factor activation. Displays weak inhibition of acetylcholinesterase, μ-opioid receptor, KCNH2 and hERG. Decreases LPI-induced GPR55 internalization. Reduces experimental intestinal inflammation in mice.

Specifications

Chemical Name or Material 4-[4,6-Dihydro-4-(3-hydroxyphenyl)-3-(4-methylphenyl)-6-oxopyrrolo[3,4-c]pyrazol-5(1H)-yl]benzoic acid
CAS 834903-43-4
Assay Percent Range >99%
Quantity 25 mg
Molecular Formula C25H19N3O4
Formula Weight Observed MW: 425.44
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