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  5. Tocris Bioscience™ CID 16020046

Tocris Bioscience™ CID 16020046
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Catalog No. 49595
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Quantity:
5 mg
25 mg
This item is not returnable. View return policy
This item is not returnable. View return policy

Description

Selective GPR55 antagonist

CID 16020046 is a selective GPR55 antagonist. Inhibits LPI-induced Ca2+ signaling (IC50 = 0.21 μM in HEK-GPR55 cells), ERK1/2 phosphorylation and GPR55-mediated transcription factor activation. Displays weak inhibition of acetylcholinesterase, μ-opioid receptor, KCNH2 and hERG. Decreases LPI-induced GPR55 internalization. Reduces experimental intestinal inflammation in mice.

Specifications

Chemical Name or Material 4-[4,6-Dihydro-4-(3-hydroxyphenyl)-3-(4-methylphenyl)-6-oxopyrrolo[3,4-c]pyrazol-5(1H)-yl]benzoic acid
CAS 834903-43-4
Assay Percent Range >99%
Quantity 5 mg
Molecular Formula C25H19N3O4
Formula Weight Observed MW: 425.44
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