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  5. Tocris Bioscience™ CP 100356 hydrochloride

Tocris Bioscience™ CP 100356 hydrochloride
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Catalog No. 419350
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Catalog No. Quantity
41-935-0 50 mg
41-931-0 10 mg
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Catalog No. 41-935-0 Supplier Tocris Bioscience™ Supplier No. 4193/50
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Description

P-gp inhibitor

High affinity P-glycoprotein (P-gp) inhibitor (Ki values are 58 and 94 nM for mouse Pgp1a and Pgp1b isoforms). Inhibits calcein-AM uptake in MDR1-transfected MDCKII cells (IC50 = 0.5 μM) and prazosin transport in BCRP-transfected MDCKII cells (IC50 = 1.5 μM). Displays weak or no inhibitory activity against MRP1, OATP1B1 and several major human P450 enzymes (IC50 > 50 μM).

Chemical Identifiers

CAS 142715-48-8
Molecular Formula C31H37ClN4O6

Specifications

Quantity 50 mg
Formula Weight 597.1
Purity >98%
Molecular Weight (g/mol) 597.109
Chemical Name or Material CP 100356 hydrochloride

Safety and Handling

Recommended Storage Desiccate at Room Temperature
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