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Tocris Bioscience™ CRT 0066101
GSA_VAGREENER_CHOICESDP

Catalog No. 497510R Shop All R&D Systems Products
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49-751-0R 10mg
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Catalog No. 49-751-0R Supplier Tocris Bioscience™ Supplier No. 4975/10
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Description

Potent protein kinase D (PKD) inhibitor

CRT 0066101 is a potent inhibitor of protein kinase D (PKD); inhibits all PKD isoforms (IC50 values are 1, 2 and 2.5 nM for PKD1, PKD3 and PKD2 respectively). Exhibits selectivity for PKD against a panel of >90 protein kinases, including PKCα, MEK, ERK, c-Raf and c-Src. Reduces proliferation and cell viability of pancreatic cancer cells expressing moderate levels of endogenous PKD1/2. Orally bioavailable.

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Specifications

Quantity 10 mg
Product Type CRT 0066101
Purity >98%
Molecular Weight (g/mol) 411.33
Inhibitors CRT 0066101

For Research Use Only

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