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  5. Tocris Bioscience™ Galeterone

Tocris Bioscience™ Galeterone
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Catalog No. 610850
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Quantity:
10 mg
50 mg
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This item is not returnable. View return policy

Description

CYP17 inhibitor; also androgen receptor antagonist

Galeterone is a CYP17 inhibitor (IC50 = 300 nM) and androgen receptor antagonist (IC50 = 384 nM in PC3-AR cells). Inhibits DHT-stimulated prostate cancer cell proliferation in vitro. Exhibits antitumor activity in SCID mice bearing prostate cancer xenografts.

Specifications

Chemical Name or Material Galeterone
CAS 851983-85-2
Synonym (3β)-17-(1H-Benzimidazol-1-yl)androsta-5,16-dien-3-ol
Quantity 50 mg
Solubility Soluble to 50mM in DMSO and to 50mM in ethanol
Molecular Formula C26H32N2O
Formula Weight 388.55
Physical Form Solid
Color White
Product Type Bioactive Small Molecule
Purity >98%
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For Research Use Only.

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