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Tocris Bioscience™ GF 109203X
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Catalog No. 07411
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Catalog No. Quantity
07-411 1 mg
07-411-0 10 mg
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Catalog No. 07-411 Supplier Tocris Bioscience™ Supplier No. 0741/1
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Description

Protein kinase C inhibitor

Very potent and selective inhibitor of protein kinase C, selective for the α and β1 isoforms (IC50 values are 0.0084, 0.0180, 0.210, 0.132, and 5.8 μM for α, β1, δ, ε and ζ isoforms respectively). Selective over MLCK, PKG and PKA (IC50 values are 0.6, 4.6, and 33 μM respectively). Potent antagonist at the 5-HT3 receptor (Ki = 29.5 nM). Anti-inflammatory in vivo.

Chemical Identifiers

CAS 133052-90-1
Molecular Formula C25H24N4O2

Specifications

Quantity 1 mg
Formula Weight 412.49
Purity >98%
Molecular Weight (g/mol) 412.493
Chemical Name or Material GF 109203X

Safety and Handling

Recommended Storage Store at Room Temperature
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