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  5. Tocris Bioscience™ GI 530159

Tocris Bioscience™ GI 530159
GREENER_CHOICE

Catalog No. 668950
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Quantity:
10 mg
50 mg
This item is not returnable. View return policy
This item is not returnable. View return policy

Description

TREK1 and TREK2 channel activator

GI 530159 is a TREK1 and TREK2 channel activator (EC50 = 0.76 μM in Rb efflux assay in TREK1-expressing CHO cells). Exhibits selectivity for TREK1/2 over TRAAK, TASK3 and a range of other potassium channels. Hyperpolarizes membrane potential of dorsal root ganglion neurons and depresses neuronal activity in vitro.

Specifications

Quantity 50 mg
Molecular Formula C27H20F6N2O2
Formula Weight 518.45
Product Type Channel Activator
Purity 99%
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