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Tocris Bioscience™ GLPG 0974
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Catalog No. 562110
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56-211-0 10 mg
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Catalog No. 56-211-0 Supplier Tocris Bioscience™ Supplier No. 5621/10
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Description

Potent FFA2 antagonist

GLPG 0974 is a potent FFA2 antagonist (IC50 = 9 nM). Exhibits selectivity for FFA2 over FFA3. Inhibits acetate-induced human neutrophil migration in plasma or buffer. Also inhibits FFA2-induced expression of CD11b activation-specific epitope (AE) in human whole blood. Orally bioavailable.

Specifications

Chemical Name or Material 4-[[[(2R)-1-(Benzo[b]thien-3-ylcarbonyl)-2-methyl-2-azetidinyl]carbonyl][(3-chlorophenyl)methyl]amino]butanoic acid
CAS 1391076-61-1
Quantity 10 mg
Target Free Fatty Acid Receptor Antagonists
Molecular Formula C25H25ClN2O4S
Formula Weight 485
Purity >98%
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