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  9. GS 6201, Tocris Bioscience™ 

GS 6201, Tocris Bioscience™ Available on GSA/VA Contract for Federal Government customers only.

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Quantity:
10mg
50mg
This item is not returnable. View return policy
752222-83-6
C21H21F3N6O2
446.434
KOYXXLLNCXWUNF-UHFFFAOYSA-N
unii-67ckv7x08g,3-ethyl-3,9-dihydro-1-propyl-8-1-3-trifluoromethyl phenyl methyl-1h-pyrazol-4-yl-1h-purine-2,6-dione,kinome_3621,d0g4cf,3-ethyl-1-propyl-8-1-3-trifluoromethyl phenyl methyl pyrazol-4-yl-7h-purine-2,6-dione,1h-purine-2,6-dione, 3-ethyl-3,9-dihydro-1-propyl-8-1-3-trifluoromethyl phenyl methyl-1h-pyrazol-4-yl,3-ethyl-1-propyl-8-1-3-trifluoromethyl benzyl-1h-pyrazol-4-yl-1h-purine-2,6 3h,7h-dione,3-ethyl-1-propyl-8-1-3-trifluoromethylbenzyl-1h-pyrazol-4-yl-3,7-dihydropurine-2,6-dione,3-ethyl-1-propyl-8-1-3-trifluoromethyl phenyl methyl pyrazol-4-yl-9h-purine-2,6-dione,8-1-3-trifluoromethyl benzyl-1h-pyrazol-4-yl-3-ethyl-1-propyl-1h-purine-2,6 3h,7h-dione
11270783
3-ethyl-1-propyl-8-[1-[[3-(trifluoromethyl)phenyl]methyl]pyrazol-4-yl]-7H-purine-2,6-dione
CCCN1C(=O)C2=C(N=C(N2)C3=CN(N=C3)CC4=CC(=CC=C4)C(F)(F)F)N(C1=O)CC
This item is not returnable. View return policy
752222-83-6
C21H21F3N6O2
446.434
KOYXXLLNCXWUNF-UHFFFAOYSA-N
unii-67ckv7x08g,3-ethyl-3,9-dihydro-1-propyl-8-1-3-trifluoromethyl phenyl methyl-1h-pyrazol-4-yl-1h-purine-2,6-dione,kinome_3621,d0g4cf,3-ethyl-1-propyl-8-1-3-trifluoromethyl phenyl methyl pyrazol-4-yl-7h-purine-2,6-dione,1h-purine-2,6-dione, 3-ethyl-3,9-dihydro-1-propyl-8-1-3-trifluoromethyl phenyl methyl-1h-pyrazol-4-yl,3-ethyl-1-propyl-8-1-3-trifluoromethyl benzyl-1h-pyrazol-4-yl-1h-purine-2,6 3h,7h-dione,3-ethyl-1-propyl-8-1-3-trifluoromethylbenzyl-1h-pyrazol-4-yl-3,7-dihydropurine-2,6-dione,3-ethyl-1-propyl-8-1-3-trifluoromethyl phenyl methyl pyrazol-4-yl-9h-purine-2,6-dione,8-1-3-trifluoromethyl benzyl-1h-pyrazol-4-yl-3-ethyl-1-propyl-1h-purine-2,6 3h,7h-dione
11270783
3-ethyl-1-propyl-8-[1-[[3-(trifluoromethyl)phenyl]methyl]pyrazol-4-yl]-7H-purine-2,6-dione
CCCN1C(=O)C2=C(N=C(N2)C3=CN(N=C3)CC4=CC(=CC=C4)C(F)(F)F)N(C1=O)CC

Description

Selective A2B antagonist

Selective antagonist of adenosine A2B receptors (Ki values are 22, 1070, 1940 and 3280 nM for human A2B, A3, A1 and A2A receptors respectively). Attenuates allergen-, NECA- and AMP-induced airway reactivity in an allergic mouse model of asthma. Also shown to attenuate the inflammatory response during acute myocardial infarction in mice; reduces caspase-1 activity in the heart.

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Quantity 10mg
Formula Weight 446.43
Percent Purity >99%
Chemical Name or Material GS 6201

Safety and Handling

Recommended Storage : Store at -20°C