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  5. Tocris Bioscience™ GSK 137647

Tocris Bioscience™ GSK 137647

Catalog No. 525710
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Quantity:
10 mg
50 mg
This item is not returnable. View return policy
This item is not returnable. View return policy

Description

Potent and selective FFA4 (GPR120) agonist

GSK 137647 is a potent and selective FFA4 (GPR120) agonist (pEC50 values are 6.3, 6.2 and 6.1 at the human, mouse and rat receptor, respectively). Exhibits ≥100-fold selectivity against a panel of 61 targets including FFA1, FFA2 and FFA3. Enhances glucose-stimulated insulin secretion in MIN6 cells. Induces intracellular calcium accumulation in U2OS cells; this activity is inhibited by AH 7614 (Cat. No. 5256).

Specifications

Purity >99%
Quantity 10 mg
Product Type GSK 137647
Molecular Weight (g/mol) 305.39
Inhibitors GSK 137647

For Research Use Only

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