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Tocris Bioscience™ GSK 429286

Catalog No. 372650R
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Catalog No. Quantity
37-265-0R 50 mg
37-261-R 1 mg
37-261-0R 10 mg
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Catalog No. 37-265-0R Supplier Tocris Bioscience™ Supplier No. 3726/50
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Description

Selective Rho-kinase (ROCK) inhibitor

GSK 429286 is a selective Rho-kinase inhibitor (IC50 values are 14, 780 and 1940 nM for ROCK1, RSK and p70S6K respectively). Reverses adrenaline-induced contraction of the rat aortic ring (IC50 = 190 nM) and causes a dose-dependent decrease in mean arterial blood pressure in spontaneous hypertensive rats. Orally active.

Specifications

Purity >97%
Gene Alias GSK429286A
Quantity 50 mg
Product Type GSK 429286
Molecular Weight (g/mol) 432.37
Inhibitors GSK 429286

For Research Use Only

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