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  5. Tocris Bioscience™ GSK 5959

Tocris Bioscience™ GSK 5959

Catalog No. 538510
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50 mg
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Catalog No. Quantity
53-851-0 10 mg
53-855-0 50 mg
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Catalog No. 53-851-0 Supplier Tocris Bioscience™ Supplier No. 5385/10
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Description

Potent and selective BRPF1 inhibitor

GSK 5959 is a potent and selective BRPF1 bromodomain inhibitor (IC50 = 80 nM). Exhibits >100-fold selectivity for BRPF1 over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. Inhibits BRPF1 interaction with histone H3.3. Cell permeable.

Specifications

Purity >99%
Quantity 10 mg
Product Type GSK 5959
Molecular Weight (g/mol) 394.47
Inhibitors GSK 5959

For Research Use Only

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