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  5. Tocris Bioscience™ GSK 626616

Tocris Bioscience™ GSK 626616
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Catalog No. 663810
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Catalog No. Quantity
66-381-0 10 mg
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Catalog No. 66-381-0 Supplier Tocris Bioscience™ Supplier No. 6638/10
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Description

Potent and selective DYRK inhibitor; orally bioavailable.

GSK 626616 is a potent and selective DYRK inhibitor (IC50 = 0.7 nM for DYRK3, similar potency for DYRK1 and 2). Exhibits ∽20-fold selectivity over casein kinase 2 and negligible activity against a panel of 451 kinases screened. Enhances number of CFU-E stimulated by Epo from human marrow. Increases hemoglobin levels in anemic mice. Orally bioavailable.

Specifications

Chemical Name or Material (5Z)-2-[(2,6-Dichlorophenyl)amino]-5-(6-quinoxalinylmethylene)-4(5H)-thiazolone
CAS 1025821-33-3
Quantity 10 mg
Molecular Formula C18H10Cl2N4OS
Formula Weight 401.27
Purity 98%
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