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  5. Tocris Bioscience™ GSK 6853

Tocris Bioscience™ GSK 6853
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Catalog No. 619825
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25 mg
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Catalog No. Quantity
61-982-5 25 mg
61-985 5 mg
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Catalog No. 61-982-5 Supplier Tocris Bioscience™ Supplier No. 6198/25
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Description

Potent and selective BRPF1 inhibitor

GSK 6853 is a potent and selective BRPF1 inhibitor. Exhibits >1600-fold selectivity for BRPF1 over other bromodomains (pIC50 values by TR-FRET are 8.1, 5.1/4.8 and 4.7/<4.3 for BRPF1, BRPF2/3 and BRD4 BD1/2, respectively).

Negative Control also available.

Specifications

Chemical Name or Material N-[2,3-dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide
CAS 1910124-24-1
Quantity 25 mg
Molecular Formula C22H27N5O3
Formula Weight 409.48
Purity 98%
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