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  5. Tocris Bioscience™ I-BRD9

Tocris Bioscience™ I-BRD9
GREENER_CHOICE

Catalog No. 559150
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Quantity:
10 mg
50 mg
This item is not returnable. View return policy
This item is not returnable. View return policy

Description

Potent and selective BRD9 inhibitor

I-BRD9 is a potent and selective BRD9 inhibitor (pIC50 = 7.3). Exhibits >70-fold selectivity for BRD9 over a panel of 34 other bromodomains and >700-fold selectivity over the BET family. Downregulates CLEC1, DUSP6, FES and SAMSN1 genes in Kasumi-1 cells.

Specifications

Chemical Name or Material 5-Ethyl-4,5-dihydro-4-oxo-N-(tetrahydro-1,1-dioxido-2H-thiopyran-4-yl)-7-[3-(trifluoromethyl)phenyl]thieno[3,2-c]pyridine-2-carboximidamide
CAS 1714146-59-4
Quantity 50 mg
Target Bromodomain Inhibitors
Molecular Formula C22H22F3N3O3S2
Formula Weight 497.55
Purity >98%
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