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Tocris Bioscience™ K 252a
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Catalog No. 1683200U Shop All R&D Systems Products
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200 μg
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Catalog No. Quantity
16-832-00U 200 μg
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Catalog No. 16-832-00U Supplier Tocris Bioscience™ Supplier No. 1683/200U
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Description

Protein kinase inhibitor

Non-selective protein kinase inhibitor; analog of staurosporine (Cat.No. 1285). Inhibits PKC (IC50 = 32.9 nM), Ca2+/calmodulin-stimulated phosphodiesterases (IC50 = 1.3 - 2.9 μM), MLCK (Ki = 20 nM) and receptor tyrosine kinases. Inhibits the oncogenic properties of MET; prevents autophosphorylation and activation of downstream effectors (MAPK, Akt).

Chemical Identifiers

CAS 99533-80-9
Molecular Formula C27H21N3O5

Specifications

Quantity 200 μg
Formula Weight 467.48
Purity >98%
Molecular Weight (g/mol) 467.481
Chemical Name or Material K 252a

Safety and Handling

Recommended Storage Desiccate at -20°C
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