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Tocris Bioscience™ Lomitapide mesylate

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Quantity:
10 mg
50 mg
Description
Lomitapide mesylate is a potent inhibitor of microsomal triglyceride transfer protein (IC50 = 8 nM). Lomitapide inhibits or normalizes lipoprotein production in rodents and in a rabbit model of hypercholesterolemia. Lomitapide is antimalarial; it inhibits hemozoin formation and growth of CQ-sensitive (PfNF54) and multidrug-resistant (PfK1) strains of P. falciparum (IC50 values are 0.56 μM and 0.69 μM respectively). Orally bioavailable.
Specifications
Specifications
Chemical Name or Material | N-(2,2,2-Trifluoroethyl)-9-[4-[4-[[[4 '-(trifluoromethyl)[1,1 '-biphenyl]-2-yl]carbonyl]amino]-1-piperidinyl]butyl]-9 H-fluorene-9-carboxamide methanesulfonate |
CAS | 2059395-52-5 |
Quantity | 50 mg |
Target | Lipid Metabolism Inhibitors |
Molecular Formula | C39H37F6N3O2.CH3SO3H |
Purity | 0.98 |
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