Tocris™ LU AA33810

Potent NPY Y5 receptor antagonist

Manufacturer: Tocris™ 3562/50

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Catalog No. 35-625-0R

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Disclaimers:

For Research Use Only


    Specifications

    Product Type LU AA33810
    Inhibitors LU AA33810
    Purity >98
    Molecular Weight 423.62
    Quantity 50mg

    Potent neuropeptide Y (NPY) Y5 receptor antagonist (Ki = 1.5nM in vitro). Displays ≥ 3300-fold affinity for Y5 over Y1, Y2 and Y4 receptors. Also binds human 5-HT2B and 5-HT1A receptors (Ki values are 247 and 478nM respectively). Exerts anxiolytic- and antidepressant-like effects in rat models of stress sensitivity.

    • Chemical Name: N-[[trans-4-[(4,5-Dihydro[1]benzothiepino[5,4-d]thiazol-2-yl)amino]cyclohexyl]methyl]methanesulfonamide
    • Formula: C19H25N3O2S3
    • CAS Number: 304008-29-5
    • Solubility: Soluble to 100mM in DMSO
    • Purity: >98

  • Description & Specifications

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