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Tocris™ MRK 740

Catalog No. 68035
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Catalog No. Quantity
68-035 5 mg
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Catalog No. 68-035 Supplier Tocris™ Supplier No. 6803/5
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Description

Potent PRDM9 inhibitor

MRK 740 is a potent PRDM9 histone methyltransferase inhibitor (IC50 = 85 nM for in vitro methylation of H3K4), which displays >100-fold selectivity over other histone methyltransferases. MRK 740 inhibits H3K4 methylation in cells (IC50 = 0.8 μM).

Specifications

Chemical Name or Material 3-(3,5-Dimethoxyphenyl)-5-(1-methyl-9-(2-methylpyridin-4-yl)-1,4,9-triazaspiro[5.5]undecan-4-yl)-1,2,4-oxadiazole
Quantity 5 mg
Molecular Formula C25H32N6O3
Purity 98%
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