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Tocris Bioscience™ PF 05190457

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Quantity:
5 mg
25 mg
Description
PF 05190457 is a high affinity and selective ghrelin receptor inverse agonist (Kd = 3 nM). Exhibits selectivity for ghrelin receptors over a panel of other targets. Increases intracellular Ca2+ concentration in and insulin secretion from human islets in vitro. Increases gastric afferent nerve activity in a rat ex vivo stomach preparation.
Specifications
Specifications
Chemical Name or Material | 1-[2-[(1R)-2,3-Dihydro-5-(6-methyl-4-pyrimidinyl)-1H-inden-1-yl]-2,7-diazaspiro[3,5]non-7-yl]-2-(2-methylimidazo[2,1-b]thiazol-6-yl)ethanone |
CAS | 1334782-79-4 |
Assay Percent Range | >98% |
Quantity | 5 mg |
Molecular Formula | C29H32N6OS |
Formula Weight | Observed MW: 512.67 |
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