R&D Systems OICR 9429, Tocris™

High affinity WDR5 antagonist

Manufacturer: R&D Systems 5267/10

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Catalog No. 526710

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Research Use Only. Not For Human or Veterinary Use


    Physical Form Solid,Solid
    Chemical Name or Material OICR 9429
    Product Type Bioactive Small Molecules
    Molecular Formula C29H32F3N5O3
    Recommended Storage Store at -20°C.
    Quantity 10mg
    Assay Percent Range >98%
    Formula Weight 555.59
    Synonym N-[2-(4-Methylpiperazin-1-yl)-5-[3-(morpholin-4-ylmethyl)phenyl]phenyl]-6-oxo-4-(trifluoromethyl)-1,6-dihydropyridine-3-carboxamide
    Solubility Soluble to 50mM in DMSO

    • Disrupts WDR5-MLL interaction
    • Exhibits selectivity for WDR5 over 22 methyltransferases and a panel of kinases, GPCRs, ion channels, and transporters
    • Reduces viability of acute myeloid leukemia cells in vitro
    • Also disrupts MLL1-RbBP5 interaction

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