Promotional price valid on web orders only. Your contract pricing may differ. Interested in signing up for a dedicated account number?
Learn More
  1. Home
  2. Products
  3. Protein Analysis Reagents
  4. Bioactive Small Molecules
  5. 787710

Tocris Bioscience™ SGC CAMKK2-1

Catalog No. 787710
Change view
Click to view available options
:
10 mg
1 product options available for selection
Product selection table with 1 available options. Use arrow keys to navigate and Enter or Space to select.
Catalog No.
78-771-0 10 mg
Use arrow keys to navigate between rows. Press Enter or Space to select a product option. 1 options available.
1 options
This item is not returnable. View return policy
Catalog No. 78-771-0 Supplier Tocris Bioscience™ Supplier No. 7877/10
Only null left
Add to Cart
Add to Cart
This item is not returnable. View return policy

Description

Potent and selective CAMKK1/2 inhibitor

SGC CAMKK2-1 is a potent and selective Ca2+-calmodulin-dependent protein kinase kinase (CaMKK) inhibitor (CAMKK2 IC50 = 30 nM). Displays selectivity toward CAMKK1 and CAMKK2 over 404 kinases in a kinome wide screen (Discoverx). SGC CAMKK2-1 inhibits AMPK phosphorylation in C4-2 prostate cancer cells (IC50 = 1.6 μM).

Specifications

Chemical Name or Material 2-Cyclopentyl-4-[5-(3-methylphenyl)furo[2,3-b]pyridin-3-yl]benzoic acid
CAS 2561494-76-4
Quantity 10 mg
Target Calcium Binding Protein Modulator Inhibitors
Molecular Formula C26H23NO3
Purity 95%
Product Title
Select an issue

By clicking Submit, you acknowledge that you may be contacted by Fisher Scientific in regards to the feedback you have provided in this form. We will not share your information for any other purposes. All contact information provided shall also be maintained in accordance with our Privacy Policy.