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  5. Tocris Bioscience™ Sitagliptin Phosphate

Tocris Bioscience™ Sitagliptin Phosphate
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Catalog No. 681610
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Catalog No. Quantity
68-161-0 10 mg
68-165-0 50 mg
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Catalog No. 68-161-0 Supplier Tocris Bioscience™ Supplier No. 6816/10
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Description

Potent and selective DPP IV (DPP4) inhibitor (IC50 = 18 nM)

Sitagliptin phosphate is a potent and selective DPP IV (DPP4) inhibitor (IC50 = 18 nM). Displays >2600-fold selectivity for DPP IV over other proline specific peptidases. Reduces blood glucose and increases GLP-1 levels after oral glucose tolerance test in normal and diet-induced obese mice.

Specifications

Chemical Name or Material (3R)-3-Amino-1-[5,6-dihydro-3-(trifluoromethyl)-1,2,4-triazolo[4,3-a]pyrazin-7(8H)-yl]-4-(2,4,5-trifluorophenyl)-1-butanone phosphate
CAS 654671-78-0
Quantity 10 mg
Molecular Formula C16H15F6N5O.H3O4P
Formula Weight 505.31
Purity 98%
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