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Tocris Bioscience™ SR 141716A

Selective CB1 receptor antagonist

Manufacturer:  Tocris Bioscience™ 0923/10

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Catalog No. 09-231-0R


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Description

Description

Potent and selective cannabinoid CB1 receptor antagonist (Ki = 1.98nM). Also acts as an inverse agonist reversing adenylyl cyclase inhibition by WIN 55,212-2 (Cat.No. 1038) (IC50 = 48nM). Displays no activity at CB2 receptors. Reduces food intake and body weight in orally dosed non-obese Wistar rats.
Specifications

Specifications

N-(Piperidin-1-yl)-5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide hydrochloride
>99%
Observed MW: 500.25
Soluble to 100mM in DMSO
158681-13-1
C22H21Cl3N4O.HCl
10mg
Safety and Handling

Safety and Handling

Recommended Storage : Desiccate at RT

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