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  5. Tocris Bioscience™ Tasimelteon

Tocris Bioscience™ Tasimelteon
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Catalog No. 749310
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Quantity:
10 mg
50 mg
This item is not returnable. View return policy
This item is not returnable. View return policy

Description

Selective dual melatonin receptor (MT1/MT2) agonist

Tasimelteon is a high affinity and selective dual melatonin receptor (MT1/MT2) agonist (Ki values are 0.304 nM and 0.0692 nM, respectively). It has no significant interaction with any other commonly screened receptors or enzyme binding sites. Tasimelteon induces a potent, concentration-dependent inhibition of forskolin-stimulated cAMP accumulation in NIH-3T3 cells stably expressing human MT1 (EC50 = 0.74 nM) or expressing human MT2 (EC50 = 0.1 nM) receptors. Tasimelteon is a circadian regulator.

Specifications

Chemical Name or Material N-[[(1 R,2 R)-2-(2,3-Dihydro-4-benzofuranyl)cyclopropyl]methyl]propanamide
CAS 609799-22-6
Quantity 10 mg
Target Melatonin (MT) Receptor Agonists
Molecular Formula C15H19NO2
Purity 0.98
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