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TCS OX2 29, Tocris Bioscience™

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Quantity:
10mg
50mg
This item is not returnable. View return policy
1610882-30-8
C23H32ClN3O3
433.977
NHKNHFJTMINMBP-ZMBIFBSDSA-N
tcs ox2 29, 2s-1-3,4-dihydro-6,7-dimethoxy-2 1h-isoquinolinyl-3,3-dimethyl-2-4-pyridinylmethyl amino-1-butanone hydrochloride, 2s-1-6,7-dimethoxy-3,4-dihydro-1h-isoquinolin-2-yl-3,3-dimethyl-2-pyridin-4-ylmethyl amino butan-1-one hydrochloride
53302033
(2S)-1-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-3,3-dimethyl-2-(pyridin-4-ylmethylamino)butan-1-one;hydrochloride
CC(C)(C)C(C(=O)N1CCC2=CC(=C(C=C2C1)OC)OC)NCC3=CC=NC=C3.Cl
This item is not returnable. View return policy
1610882-30-8
C23H32ClN3O3
433.977
NHKNHFJTMINMBP-ZMBIFBSDSA-N
tcs ox2 29, 2s-1-3,4-dihydro-6,7-dimethoxy-2 1h-isoquinolinyl-3,3-dimethyl-2-4-pyridinylmethyl amino-1-butanone hydrochloride, 2s-1-6,7-dimethoxy-3,4-dihydro-1h-isoquinolin-2-yl-3,3-dimethyl-2-pyridin-4-ylmethyl amino butan-1-one hydrochloride
53302033
(2S)-1-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-3,3-dimethyl-2-(pyridin-4-ylmethylamino)butan-1-one;hydrochloride
CC(C)(C)C(C(=O)N1CCC2=CC(=C(C=C2C1)OC)OC)NCC3=CC=NC=C3.Cl

Potent and selective OX2 antagonist

Potent and selective OX2 receptor antagonist (IC50 = 40 nM). Displays >250-fold selectivity for OX2 over OX1 and a range of receptors, ion channels and transporters. Inhibits orexin A induced IP3 accumulation and ERK1/2 phosphorylation in CHO cells transfected with the OX2 receptor.
Quantity 10mg
Formula Weight 433.97
Percent Purity >98%
Chemical Name or Material TCS OX2 29

Recommended Storage : Desiccate at +4°C