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Tocris Bioscience™ VU 0463271
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Catalog No. 471950
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47-195-0 50 mg
47-191-0 10 mg
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Catalog No. 47-195-0 Supplier Tocris Bioscience™ Supplier No. 4719/50
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Description

Potent and selective KCC2 inhibitor

VU 0463271 is a potent and selective inhibitor of the neuronal K-Cl cotransporter, KCC2 (IC50 = 61 nM); displays >100-fold selectivity versus the Na-K-2Cl cotransporter 1 (NKCC1) and no activity against a panel of 68 GPCRs, ion channels and transporters.

Specifications

Chemical Name or Material N-Cyclopropyl-N-(4-methyl-2-thiazolyl)-2-[(6-phenyl-3-pyridazinyl)thio]acetamide
CAS 1391737-01-1
Quantity 50 mg
Target KCC2 Inhibitors
Molecular Formula C19H18N4OS2
Formula Weight 382.5
Purity >98%
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